| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50082313 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_209602 |
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| Ki | 625±n/a nM |
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| Citation |  Halmos, T; Turek, JW; Le Breton, GC; Antonakis, K Synthesis and biological characterization of sqbazide, a novel biotinylated photoaffinity probe for the study of the human platelet thromboxane A2 receptor. Bioorg Med Chem Lett9:2963-8 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50082313 |
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| n/a |
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| Name | BDBM50082313 |
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| Synonyms: | 4-(4-Azido-phenyl)-N-({[3-((Z)-7-oxo-7-{N'-[5-((3aS,6R,6aR)-2-oxo-hexahydro-thieno[3,4-d]imidazol-6-yl)-pentanoyl]-hydrazino}-hept-2-enyl)-7-oxa-bicyclo[2.2.1]hept-2-ylmethyl]-carbamoyl}-methyl)-butyramide | CHEMBL99695 |
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| Type | Small organic molecule |
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| Emp. Form. | C36H51N9O6S |
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| Mol. Mass. | 737.912 |
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| SMILES | [N-]=[N+]=Nc1ccc(CCCC(=O)NCC(=O)NCC2C3CCC(O3)C2C\C=C/CCCC(=O)NNC(=O)CCCC[C@H]2SC[C@H]3NC(=O)N[C@@H]23)cc1 |TLB:25:24:23:20.21,THB:17:18:23:20.21| |
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| Structure | 
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