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TargetChymotrypsin-like elastase family member 2A
LigandBDBM50089099
Substrate/Competitorn/a
Meas. Tech.ChEBML_152317
Ki 1100000±n/a nM
Citation Wright, PARostom, AARobinson, CVSchofield, CJ Mass spectrometry reveals elastase inhibitors from the reactive centre loop of alpha1-antitrypsin. Bioorg Med Chem Lett10:1219-21 (2000) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Chymotrypsin-like elastase family member 2A
Name:Chymotrypsin-like elastase family member 2A
Synonyms:CEL2A_PIG | CELA2A | ELA2 | ELA2A | Elastase 2A | Elastase-2 | Elastase-2A | Pancreatic elastase
Type:PROTEIN
Mol. Mass.:28705.23
Organism:Sus scrofa
Description:ChEMBL_156951
Residue:269
Sequence:
MIRALLLSTLVAGALSCGLPANLPQLPRVVGGEDARPNSWPWQVSLQYDSSGQWRHTCGG
TLVDQSWVLTAAHCISSSRTYRVVLGRHSLSTNEPGSLAVKVSKLVVHQDWNSNQLSNGN
DIALLKLASPVSLTDKIQLGCLPAAGTILPNNYVCYVTGWGRLQTNGASPDILQQGQLLV
VDYATCSKPGWWGSTVKTNMICAGGDGIISSCNGDSGGPLNCQGANGQWQVHGIVSFGSS
LGCNYYHKPSVFTRVSNYIDWINSVIANN
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  Blast E-value cutoff:
BDBM50089099
n/a
NameBDBM50089099
Synonyms:(S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-methylsulfanyl-butyrylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-propionic acid | CHEMBL20112
TypeSmall organic molecule
Emp. Form.C23H36N4O5S
Mol. Mass.480.621
SMILESCSCC[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(O)=O
Structure
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