| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50092588 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_46458 (CHEMBL657905) |
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| Ki | 33±n/a nM |
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| Citation |  Mahadevan, A; Siegel, C; Martin, BR; Abood, ME; Beletskaya, I; Razdan, RK Novel cannabinol probes for CB1 and CB2 cannabinoid receptors. J Med Chem43:3778-85 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52868.96 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21554 |
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| Residue: | 472 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50092588 |
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| n/a |
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| Name | BDBM50092588 |
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| Synonyms: | 4-(1,1-Dimethyl-heptyl)-2'-isopropyl-5'-methyl-biphenyl-2-ol | CHEMBL125061 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H36O |
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| Mol. Mass. | 352.5527 |
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| SMILES | CCCCCCC(C)(C)c1ccc(c(O)c1)-c1cc(C)ccc1C(C)C |
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| Structure | 
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