| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 1E |
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| Ligand | BDBM34141 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_2052 |
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| Ki | 4220.0±n/a nM |
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| Citation |  Tsai, Y; Dukat, M; Slassi, A; MacLean, N; Demchyshyn, L; Savage, JE; Roth, BL; Hufesein, S; Lee, M; Glennon, RA N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists. Bioorg Med Chem Lett10:2295-9 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 1E |
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| Name: | 5-hydroxytryptamine receptor 1E |
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| Synonyms: | 5-HT-1E | 5-HT1E | 5-Hydroxytryptamine Receptor Subtype 1E (5HT1E) | 5-hydroxytryptamine receptor 1E | 5-hydroxytryptamine receptor 1E (5-HT-1E) (S31) | 5-hydroxytryptamine receptor 1E (5-HT-1E) (Serotonin receptor 1E) (5-HT1E) (S31). | 5HT1E_HUMAN | HTR1E | S31 | Serotonin (5-HT) receptor | Serotonin 1e (5-HT1e) receptor | Serotonin Receptor 1E |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 41697.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_112822 |
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| Residue: | 365 |
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| Sequence: | MNITNCTTEASMAIRPKTITEKMLICMTLVVITTLTTLLNLAVIMAIGTTKKLHQPANYL
ICSLAVTDLLVAVLVMPLSIIYIVMDRWKLGYFLCEVWLSVDMTCCTCSILHLCVIALDR
YWAITNAIEYARKRTAKRAALMILTVWTISIFISMPPLFWRSHRRLSPPPSQCTIQHDHV
IYTIYSTLGAFYIPLTLILILYYRIYHAAKSLYQKRGSSRHLSNRSTDSQNSFASCKLTQ
TFCVSDFSTSDPTTEFEKFHASIRIPPFDNDLDHPGERQQISSTRERKAARILGLILGAF
ILSWLPFFIKELIVGLSIYTVSSEVADFLTWLGYVNSLINPLLYTSFNEDFKLAFKKLIR
CREHT
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| BDBM34141 |
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| n/a |
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| Name | BDBM34141 |
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| Synonyms: | CHEMBL76237 | MS-245 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22N2O3S |
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| Mol. Mass. | 358.455 |
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| SMILES | COc1ccc2n(cc(CCN(C)C)c2c1)S(=O)(=O)c1ccccc1 |
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| Structure | 
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