| Reaction Details |
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 | Report a problem with these data |
| Target | Histamine H3 receptor |
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| Ligand | BDBM50098205 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_86751 |
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| Ki | 44±n/a nM |
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| Citation |  Stark, H; Sippl, W; Ligneau, X; Arrang, JM; Ganellin, CR; Schwartz, JC; Schunack, W Different antagonist binding properties of human and rat histamine H3 receptors. Bioorg Med Chem Lett11:951-4 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Histamine H3 receptor |
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| Name: | Histamine H3 receptor |
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| Synonyms: | HH3R | HRH3_RAT | Hrh3 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 48607.98 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 445 |
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| Sequence: | MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFV
ADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCAS
SVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGG
SSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAG
PEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRYGVGEAGPGVEAGEAALGGGSGGGAA
ASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSL
AIIVSIFGLCWAPYTLLMIIRAACHGRCIPDYWYETSFWLLWANSAVNPVLYPLCHYSFR
RAFTKLLCPQKLKVQPHGSLEQCWK
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| BDBM50098205 |
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| n/a |
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| Name | BDBM50098205 |
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| Synonyms: | 1-{4-[3-(1H-Imidazol-4-yl)-propylsulfanyl]-phenyl}-ethanone | CHEMBL424365 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H16N2OS |
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| Mol. Mass. | 260.355 |
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| SMILES | CC(=O)c1ccc(SCCCc2cnc[nH]2)cc1 |
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| Structure | 
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