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TargetSomatostatin receptor type 4
LigandBDBM50098605
Substrate/Competitorn/a
Meas. Tech.ChEMBL_200840 (CHEMBL807050)
Kd 1000±n/a nM
Citation Rajeswaran, WG; Hocart, SJ; Murphy, WA; Taylor, JE; Coy, DH N-Methyl scan of somatostatin octapeptide agonists produces interesting effects on receptor subtype specificity. J Med Chem44:1416-21 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Somatostatin receptor type 4
Name:Somatostatin receptor type 4
Synonyms:SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4)
Type:Enzyme
Mol. Mass.:42015.38
Organism:Homo sapiens (Human)
Description:P31391
Residue:388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
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BDBM50098605
n/a
NameBDBM50098605
Synonyms:10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl)-propionylamino]-16-benzyl-7-(1-hydroxy-ethyl)-13-(1H-indol-3-ylmethyl)-8-methyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carboxylic acid (1-carbamoyl-2-hydroxy-propyl)-amide | CHEMBL437093
TypeSmall organic molecule
Emp. Form.C50H67N11O11S2
Mol. Mass.1062.264
SMILESC[C@@H](O)[C@H](NC(=O)[C@@H]1CSSC[C@@H](NC(=O)[C@H](N)Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N(C)[C@@H]([C@@H](C)O)C(=O)N1)C(N)=O
Structure
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