| Reaction Details |
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 | Report a problem with these data |
| Target | Carnitine O-palmitoyltransferase 1, muscle isoform |
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| Ligand | BDBM50101593 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_46323 (CHEMBL660891) |
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| IC50 | 211000±n/a nM |
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| Citation |  Giannessi, F; Chiodi, P; Marzi, M; Minetti, P; Pessotto, P; De Angelis, F; Tassoni, E; Conti, R; Giorgi, F; Mabilia, M; Dell'Uomo, N; Muck, S; Tinti, MO; Carminati, P; Arduini, A Reversible carnitine palmitoyltransferase inhibitors with broad chemical diversity as potential antidiabetic agents. J Med Chem44:2383-6 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Carnitine O-palmitoyltransferase 1, muscle isoform |
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| Name: | Carnitine O-palmitoyltransferase 1, muscle isoform |
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| Synonyms: | CPT1B_RAT | Carnitine palmitoyltransferase 1B | Cpt1b |
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| Type: | PROTEIN |
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| Mol. Mass.: | 88241.28 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_887447 |
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| Residue: | 772 |
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| Sequence: | MAEAHQAVAFQFTVTPDGVDFRLSREALRHIYLSGINSWKKRLIRIKNGILRGVYPGSPT
SWLVVVMATVGSNYCKVDISMGLVHCIQRCLPTRYGSYGTPQTETLLSMVIFSTGVWATG
IFLFRQTLKLLLSYHGWMFEMHSKTSHATKIWAICVRLLSSRRPMLYSFQTSLPKLPVPS
VPATIHRYLDSVRPLLDDEAYFRMESLAKEFQDKIAPRLQKYLVLKSWWATNYVSDWWEE
YVYLRGRSPIMVNSNYYAMDFVLIKNTSQQAARLGNTVHAMIMYRRKLDREEIKPVMALG
MVPMCSYQMERMFNTTRIPGKETDLLQHLSESRHVAVYHKGRFFKVWLYEGSCLLKPRDL
EMQFQRILDDTSPPQPGEEKLAALTAGGRVEWAEARQKFFSSGKNKMSLDTIERAAFFVA
LDEDSHCYNPDDEASLSLYGKSLLHGNCYNRWFDKSFTLISCKNGQLGLNTEHSWADAPI
IGHLWEFVLATDTFHLGYTETGHCVGEPNTKLPPPQRMQWDIPEQCQTAIENSYQVAKAL
ADDVELYCFQFLPFGKGLIKKCRTSPDAFVQIALQLAHFRDKGKFCLTYEASMTRMFREG
RTETVRSCTSESTAFVRAMMTGSHKKQDLQDLFRKASEKHQNMYRLAMTGAGIDRHLFCL
YIVSKYLGVRSPFLDEVLSEPWSLSTSQIPQFQICMFDPKQYPNHLGAGGGFGPVADHGY
GVSYMIAGENTMFFHVSSKLSSSETNALRFGNHIRQALLDIADLFKISKTDS
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| BDBM50101593 |
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| n/a |
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| Name | BDBM50101593 |
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| Synonyms: | (3-Carboxy-2-octyloxycarbonylamino-propyl)-trimethyl-ammonium | CHEMBL78979 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H32N2O4 |
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| Mol. Mass. | 316.4363 |
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| SMILES | CCCCCCCCOC(=O)NC(CC([O-])=O)C[N+](C)(C)C |
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| Structure | 
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