| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM50101787 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_29638 |
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| Ki | 18±n/a nM |
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| Citation |  van Tilburg, EW; van der Klein, PA; de Groote, M; Beukers, MW; IJzerman, AP Substituted 4-phenyl-2-(phenylcarboxamido)-1,3-thiazole derivatives as antagonists for the adenosine A(1) receptor. Bioorg Med Chem Lett11:2017-9 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM50101787 |
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| n/a |
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| Name | BDBM50101787 |
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| Synonyms: | 4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEMBL62078 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H11ClN2OS |
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| Mol. Mass. | 314.789 |
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| SMILES | Clc1ccc(cc1)C(=O)Nc1nc(cs1)-c1ccccc1 |
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| Structure | 
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