| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50097423 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_29903 |
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| Ki | 82±n/a nM |
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| Citation |  van Tilburg, EW; van der Klein, PA; de Groote, M; Beukers, MW; IJzerman, AP Substituted 4-phenyl-2-(phenylcarboxamido)-1,3-thiazole derivatives as antagonists for the adenosine A(1) receptor. Bioorg Med Chem Lett11:2017-9 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM50097423 |
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| n/a |
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| Name | BDBM50097423 |
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| Synonyms: | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzamide | 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzamide(LUF5417) | 4-methoxy-N-(3-phenyl-1,2,4-thiadiazol-5-yl)benzamide | CHEMBL305322 | LUF-5417 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13N3O2S |
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| Mol. Mass. | 311.358 |
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| SMILES | COc1ccc(cc1)C(=O)Nc1nc(ns1)-c1ccccc1 |
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| Structure | 
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