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TargetProstanoid EP2 receptor
LigandBDBM50101823
Substrate/Competitorn/a
Meas. Tech.ChEMBL_158309
Ki 25±n/a nM
Citation Tani KNaganawa AIshida AEgashira HSagawa KHarada HOgawa MMaruyama TOhuchida SNakai HKondo KToda M Design and synthesis of a highly selective EP2-receptor agonist. Bioorg Med Chem Lett 11:2025-8 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Prostanoid EP2 receptor
Name:Prostanoid EP2 receptor
Synonyms:PGE receptor, EP2 subtype | Prostaglandin E2 | Prostaglandin E2 receptor EP2 subtype
Type:G-protein coupled receptor
Mol. Mass.:40495.26
Organism:Mus musculus (Mouse)
Description:n/a
Residue:362
Sequence:
MDNFLNDSKLMEDCKSRQWLLSGESPAISSVMFSAGVLGNLIALALLARRWRGDTGCSAG
SRTSISLFHVLVTELVLTDLLGTCLISPVVLASYSRNQTLVALAPESHACTYFAFTMTFF
SLATMLMLFAMALERYLSIGYPYFYRRHLSRRGGLAVLPVIYGASLLFCSLPLLNYGEYV
QYCPGTWCFIRHGRTAYLQLYATMLLLLIVAVLACNISVILNLIRMHRRSRRSRCGLSGS
SLRGPGSRRRGERTSMAEETDHLILLAIMTITFAICSLPFTIFAYMDETSSLKEKWDLRA
LRFLSVNSIIDPWVFAILRPPVLRLMRSVLCCRTSLRTQEAQQTSCSTQSSASKQTDLCG
QL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50101823
n/a
NameBDBM50101823
Synonyms:4-(2-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-ethyl)-benzoic acid | CHEMBL64423
TypeSmall organic molecule
Emp. Form.C25H34O5
Mol. Mass.414.5345
SMILESCCCC1(CCC1)[C@@H](O)C\C=C\C1[C@H](O)CC(=O)[C@@H]1CCc1ccc(cc1)C(O)=O
Structure
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