| Reaction Details |
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 | Report a problem with these data |
| Target | Prostanoid EP4 Receptor |
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| Ligand | BDBM50101822 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_158449 |
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| Ki | 3.1±n/a nM |
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| Citation |  Tani K; Naganawa A; Ishida A; Egashira H; Sagawa K; Harada H; Ogawa M; Maruyama T; Ohuchida S; Nakai H; Kondo K; Toda M Design and synthesis of a highly selective EP2-receptor agonist. Bioorg Med Chem Lett 11:2025-8 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostanoid EP4 Receptor |
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| Name: | Prostanoid EP4 receptor |
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| Synonyms: | PGE receptor, EP4 subtype |
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| Type: | G-protein coupled receptor |
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| Mol. Mass.: | 56175.66 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | n/a |
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| Residue: | 513 |
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| Sequence: | MAEVGGTIPRSNRELQRCVLLTTTIMSIPGVNASFSSTPERLNSPVTIPAVMFIFGVVGN
LVAIVVLCKSRKEQKETTFYTLVCGLAVTDLLGTLLVSPVTIATYMKGQWPGDQALCDYS
TFILLFFGLSGLSIICAMSIERYLAINHAYFYSHYVDKRLAGLTLFAIYASNVLFCALPN
MGLGRSERQYPGTWCFIDWTTNVTAYAAFSYMYAGFSSFLILATVLCNVLVCGALLRMHR
QFMRRTSLGTEQHHAAAAAAVASVACRGHAGASPALQRLSDFRRRRSFRRIAGAEIQMVI
LLIATSLVVLICSIPLVVRVFINQLYQPNVVKDISRNPDLQAIRIASVNPILDPWIYILL
RKTVLSKAIEKIKCLFCRIGGSGRDSSAQHCSESRRTSSAMSGHSRSFLARELKEISSTS
QTLLYLPDLTESSLGGRNLLPGSHGMGLTQADTTSLRTLRISETSDSSQGQDSESVLLVD
EVSGSHREEPASKGNSLQVTFPSETLKLSEKCI
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| BDBM50101822 |
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| n/a |
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| Name | BDBM50101822 |
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| Synonyms: | (Z)-7-[(1R,2R,3R)-3-Hydroxy-2-((E)-(R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-hept-5-enoic acid | CHEMBL64804 | PGE2, 15-epi | US9180116, PGE2 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H32O5 |
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| Mol. Mass. | 352.4651 |
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| SMILES | CCCCC[C@@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1C\C=C/CCCC(O)=O |
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| Structure | 
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