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TargetProstaglandin E2 receptor EP1 subtype
LigandBDBM50101819
Substrate/Competitorn/a
Meas. Tech.ChEBML_158179
Ki 780±n/a nM
Citation Tani, KNaganawa, AIshida, AEgashira, HSagawa, KHarada, HOgawa, MMaruyama, TOhuchida, SNakai, HKondo, KToda, M Design and synthesis of a highly selective EP2-receptor agonist. Bioorg Med Chem Lett11:2025-8 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Prostaglandin E2 receptor EP1 subtype
Name:Prostaglandin E2 receptor EP1 subtype
Synonyms:PE2R1_MOUSE | PGE receptor, EP1 subtype | Prostaglandin E1 | Prostaglandin E2 receptor EP1 subtype | Prostanoid EP1 receptor | Ptger1 | Ptgerep1
Type:G-protein coupled receptor
Mol. Mass.:43000.62
Organism:Mus musculus (Mouse)
Description:n/a
Residue:405
Sequence:
MSPCGLNLSLADEAATCATPRLPNTSVVLPTGDNGTSPALPIFSMTLGAVSNVLALALLA
QVAGRMRRRRSAATFLLFVASLLAIDLAGHVIPGALVLRLYTAGRAPAGGACHFLGGCMV
FFGLCPLLLGCGMAVERCVGVTQPLIHAARVSVARARLALAVLAAMALAVALLPLVHVGR
YELQYPGTWCFISLGPRGGWRQALLAGLFAGLGLAALLAALVCNTLSGLALLRARWRRRR
SRRFRKTAGPDDRRRWGSRGPRLASASSASSITSATATLRSSRGGGSARRVHAHDVEMVG
QLVGIMVVSCICWSPLLVLVVLAIGGWNSNSLQRPLFLAVRLASWNQILDPWVYILLRQA
MLRQLLRLLPLRVSAKGGPTELGLTKSAWEASSLRSSRHSGFSHL
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  Blast E-value cutoff:
BDBM50101819
n/a
NameBDBM50101819
Synonyms:(Z)-7-{(1R,2R,3R)-2-[(E)-(S)-4-(1-Butyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-5-oxo-cyclopentyl}-hept-5-enoic acid | CHEMBL303763
TypeSmall organic molecule
Emp. Form.C24H38O5
Mol. Mass.406.5555
SMILESCCCCC1(CCC1)[C@@H](O)C\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1C\C=C/CCCC(O)=O
Structure
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