| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM50109386 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_201564 |
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| Ki | 5.9±n/a nM |
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| Citation |  Maeda, DY; Williams, W; Kim, WE; Thatcher, LN; Bowen, WD; Coop, A N-arylalkylpiperidines as high-affinity sigma-1 and sigma-2 receptor ligands: phenylpropylamines as potential leads for selective sigma-2 agents. Bioorg Med Chem Lett12:497-500 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25266.54 |
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| Organism: | RAT |
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| Description: | Q9R0C9 |
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| Residue: | 223 |
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| Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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| BDBM50109386 |
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| n/a |
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| Name | BDBM50109386 |
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| Synonyms: | 2-Phenethyl-1,2,3,4-tetrahydro-isoquinoline | CHEMBL146238 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H19N |
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| Mol. Mass. | 237.3395 |
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| SMILES | C(Cc1ccccc1)N1CCc2ccccc2C1 |
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| Structure | 
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