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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50109389
Substrate/Competitorn/a
Meas. Tech.ChEBML_201564
Ki 89±n/a nM
Citation Maeda, DYWilliams, WKim, WEThatcher, LNBowen, WDCoop, A N-arylalkylpiperidines as high-affinity sigma-1 and sigma-2 receptor ligands: phenylpropylamines as potential leads for selective sigma-2 agents. Bioorg Med Chem Lett12:497-500 (2002) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1
Type:Enzyme Catalytic Domain
Mol. Mass.:25266.54
Organism:RAT
Description:Q9R0C9
Residue:223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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  Blast E-value cutoff:
BDBM50109389
n/a
NameBDBM50109389
Synonyms:1-Phenethyl-piperidine | 1-phenethylpiperidine | CHEMBL75228 | N-(2-phenylethyl)piperidine | N-phenethylpiperidine
TypeSmall organic molecule
Emp. Form.C13H19N
Mol. Mass.189.2967
SMILESC(Cc1ccccc1)N1CCCCC1
Structure
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