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TargetCannabinoid receptor 1
LigandBDBM50117179
Substrate/Competitorn/a
Meas. Tech.ChEMBL_46465
Ki 389±n/a nM
Citation Barnett-Norris JHurst DPLynch DLGuarnieri FMakriyannis AReggio PH Conformational memories and the endocannabinoid binding site at the cannabinoid CB1 receptor. J Med Chem 45:3649-59 (2002) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 1
Name:Cannabinoid receptor 1
Synonyms:CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain)
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:52868.96
Organism:Homo sapiens (Human)
Description:P21554
Residue:472
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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  Blast E-value cutoff:
BDBM50117179
n/a
NameBDBM50117179
Synonyms:1N-[2-hydroxy-1-methyl-(1S)-ethyl]-2-methyl-(2S,5Z,8Z,11Z,14Z)-5,8,11,14-icosatetraenamide | CHEMBL120105
TypeSmall organic molecule
Emp. Form.C24H41NO2
Mol. Mass.375.5878
SMILESCCCCC\C=C/C\C=C/C\C=C/C\C=C/CC[C@H](C)C(=O)N[C@@H](C)CO
Structure
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