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TargetPlatelet-activating factor receptor
LigandBDBM50118194
Substrate/Competitorn/a
Meas. Tech.ChEMBL_155144 (CHEMBL760185)
Ki 150±n/a nM
Citation Strømgaard, KSaito, DRShindou, HIshii, SShimizu, TNakanishi, K Ginkgolide derivatives for photolabeling studies: preparation and pharmacological evaluation. J Med Chem45:4038-46 (2002) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Platelet-activating factor receptor
Name:Platelet-activating factor receptor
Synonyms:PAF-R | PTAFR_MOUSE | Platelet activating factor receptor | Platelet-activating factor receptor | Ptafr
Type:PROTEIN
Mol. Mass.:39163.36
Organism:Mus musculus
Description:ChEMBL_155144
Residue:341
Sequence:
MEHNGSFRVDSEFRYTLFPIVYSVIFILGVVANGYVLWVFANLYPSKKLNEIKIFMVNLT
MADLLFLITLPLWIVYYYNEGDWILPNFLCNVAGCLFFINTYCSVAFLGVITYNRYQAVA
YPIKTAQATTRKRGISLSLIIWVSIVATASYFLATDSTNLVPNKDGSGNITRCFEHYEPY
SVPILVVHVFIAFCFFLVFFLIFYCNLVIIHTLLTQPMRQQRKAGVKRRALWMVCTVLAV
FIICFVPHHVVQLPWTLAELGYQTNFHQAINDAHQITLCLLSTNCVLDPVIYCFLTKKFR
KHLSEKFYSMRSSRKCSRATSDTCTEVIVPANQTPIVSLKN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50118194
n/a
NameBDBM50118194
Synonyms:8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-trifluoromethyl-3H-1,2-diaziren-3-yl)benzyloxy]-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | CHEMBL339146
TypeSmall organic molecule
Emp. Form.C29H29F3N2O10
Mol. Mass.622.5432
SMILESn/a
Structure
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