| Reaction Details |
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 | Report a problem with these data |
| Target | Peroxisome proliferator-activated receptor gamma |
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| Ligand | BDBM50121412 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_154362 |
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| Ki | 2200±n/a nM |
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| Citation |  Thor, M; Beierlein, K; Dykes, G; Gustavsson, AL; Heidrich, J; Jendeberg, L; Lindqvist, B; Pegurier, C; Roussel, P; Slater, M; Svensson, S; Sydow-Bäckman, M; Thornström, U; Uppenberg, J Synthesis and pharmacological evaluation of a new class of peroxisome proliferator-activated receptor modulators. Bioorg Med Chem Lett12:3565-7 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Peroxisome proliferator-activated receptor gamma |
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| Name: | Peroxisome proliferator-activated receptor gamma |
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| Synonyms: | NR1C3 | Nuclear receptor subfamily 1 group C member 3 | PPAR-gamma | PPARG | PPARG_HUMAN | Peroxisome proliferator-activated receptor | Peroxisome proliferator-activated receptor gamma (PPAR gamma) | Peroxisome proliferator-activated receptor gamma (PPARG) | Peroxisome proliferator-activated receptor gamma (PPARĪ³) | Peroxisome proliferator-activated receptor gamma/Nuclear receptor corepressor 2 | peroxisome proliferator-activated receptor gamma isoform 2 |
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| Type: | Nuclear Receptor |
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| Mol. Mass.: | 57613.46 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P37231 |
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| Residue: | 505 |
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| Sequence: | MGETLGDSPIDPESDSFTDTLSANISQEMTMVDTEMPFWPTNFGISSVDLSVMEDHSHSF
DIKPFTTVDFSSISTPHYEDIPFTRTDPVVADYKYDLKLQEYQSAIKVEPASPPYYSEKT
QLYNKPHEEPSNSLMAIECRVCGDKASGFHYGVHACEGCKGFFRRTIRLKLIYDRCDLNC
RIHKKSRNKCQYCRFQKCLAVGMSHNAIRFGRMPQAEKEKLLAEISSDIDQLNPESADLR
ALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQE
QSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLAS
LMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVII
LSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQL
LQVIKKTETDMSLHPLLQEIYKDLY
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| BDBM50121412 |
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| n/a |
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| Name | BDBM50121412 |
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| Synonyms: | 2-(2,4-Dichloro-benzoylamino)-5-methyl-benzoic acid | CHEMBL118972 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H11Cl2NO3 |
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| Mol. Mass. | 324.159 |
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| SMILES | Cc1ccc(NC(=O)c2ccc(Cl)cc2Cl)c(c1)C(O)=O |
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| Structure | 
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