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TargetMu-type opioid receptor
LigandBDBM50124002
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145281 (CHEMBL751217)
Ki 3.6±n/a nM
Citation Wentland, MPYe, YCioffi, CLLou, RZhou, QXu, GDuan, WDehnhardt, CMSun, XCohen, DJBidlack, JM Syntheses and opioid receptor binding affinities of 8-amino-2,6-methano-3-benzazocines. J Med Chem46:838-49 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50124002
n/a
NameBDBM50124002
Synonyms:8-Amino-3-cyclopropylmethyl-6,11-dimethyl-3,4,5,6-tetrahydro-2H-2,6-methano-benzo[d]azocin-1-one | CHEMBL422560
TypeSmall organic molecule
Emp. Form.C18H24N2O
Mol. Mass.284.396
SMILESC[C@H]1C2N(CC3CC3)CC[C@]1(C)c1cc(N)ccc1C2=O |TLB:4:3:19.12.18:1,13:12:1:3.9.8,THB:20:19:1:3.9.8|
Structure
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