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TargetMu-type opioid receptor
LigandBDBM50085023
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145281 (CHEMBL751217)
Ki 9±n/a nM
Citation Wentland, MPYe, YCioffi, CLLou, RZhou, QXu, GDuan, WDehnhardt, CMSun, XCohen, DJBidlack, JM Syntheses and opioid receptor binding affinities of 8-amino-2,6-methano-3-benzazocines. J Med Chem46:838-49 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50085023
n/a
NameBDBM50085023
Synonyms:((6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-yl)-phenethyl-amine | (3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-yl)-phenethyl-amine | CHEMBL56165
TypeSmall organic molecule
Emp. Form.C26H34N2
Mol. Mass.374.5616
SMILESC[C@H]1C2Cc3ccc(NCCc4ccccc4)cc3[C@@]1(C)CCN2CC1CC1 |TLB:24:23:1:18.4.3,17:18:1:23.21.22|
Structure
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