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TargetNeuropeptide Y receptor type 5 ( NPY Y5)
LigandBDBM50128936
Substrate/Competitorn/a
Meas. Tech.ChEBML_144128
Ki 15±n/a nM
Citation Hammond MElliott RLGillaspy MLHager DCHank RFLaFlamme JAOliver RMDaSilva-Jardine PAStevenson RWMack CMCassella JV Structure-activity relationships in a series of NPY Y5 antagonists: 3-amido-9-ethylcarbazoles, core-modified analogues and amide isosteres. Bioorg Med Chem Lett 13:1989-92 (2003) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Neuropeptide Y receptor type 5 ( NPY Y5)
Name:Neuropeptide Y receptor type 5
Synonyms:NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPYY5 | Y5 receptor
Type:Enzyme
Mol. Mass.:50746.64
Organism:Homo sapiens (Human)
Description:Q15761
Residue:445
Sequence:
MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNL
LILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFL
QCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSL
VELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISC
GLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAP
ERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIK
KRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCL
NPILYGFLNNGIKADLVSLIHCLHM
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  Blast E-value cutoff:
BDBM50128936
n/a
NameBDBM50128936
Synonyms:2,2,2-Trifluoro-N-(9-isopropyl-9H-carbazol-3-yl)-acetamide | CHEMBL294842
TypeSmall organic molecule
Emp. Form.C17H15F3N2O
Mol. Mass.320.309
SMILESCC(C)n1c2ccccc2c2cc(NC(=O)C(F)(F)F)ccc12
Structure
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