| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 5A |
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| Ligand | BDBM50132129 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_3595 (CHEMBL618080) |
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| Ki | 130±n/a nM |
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| Citation |  Khorana, N; Smith, C; Herrick-Davis, K; Purohit, A; Teitler, M; Grella, B; Dukat, M; Glennon, RA Binding of tetrahydrocarboline derivatives at human 5-HT5A receptors. J Med Chem46:3930-7 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 5A |
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| Name: | 5-hydroxytryptamine receptor 5A |
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| Synonyms: | 5-HT-5 | 5-HT-5A | 5-HT5 | 5-HT5a | 5-hydroxytryptamine receptor 5A | 5HT5A_MOUSE | 5ht5a | Htr5a | Serotonin 5a (5-HT5a) receptor | Serotonin receptor 5A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40749.33 |
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| Organism: | MOUSE |
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| Description: | 5-HT5 0 MOUSE::P30966 |
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| Residue: | 357 |
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| Sequence: | MDLPVNLTSFSLSTPSSLEPNRSLDTEVLRPSRPFLSAFRVLVLTLLGFLAAATFTWNLL
VLATILKVRTFHRVPHNLVASMAISDVLVAVLVMPLSLVHELSGRRWQLGRRLCQLWIAC
DVLCCTASIWNVTAIALDRYWSITRHLEYTLRTRKRVSNVMILLTWALSTVISLAPLLFG
WGETYSEPSEECQVSREPSYTVFSTVGAFYLPLCVVLFVYWKIYRAAKFRMGSRKTNSVS
PVPEAVEVKNATQHPQMVFTVRHATVTFQTEGDTWREQKEQRAALMVGILIGVFVLCWFP
FFVTELISPLCSWDVPAIWKSIFLWLGYSNSFFNPLIYTAFNRSYSSAFKVFFSKQQ
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| BDBM50132129 |
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| n/a |
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| Name | BDBM50132129 |
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| Synonyms: | 5-Methyl-2-(4-phenyl-butyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole | CHEMBL129472 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H26N2 |
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| Mol. Mass. | 318.4552 |
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| SMILES | Cn1c2CCN(CCCCc3ccccc3)Cc2c2ccccc12 |
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| Structure | 
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