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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Carboxypeptidase M | ||
| Ligand | BDBM50135939 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_45790 | ||
| IC50 | 13±n/a nM | ||
| Citation |  Barrow JC; Nantermet PG; Stauffer SR; Ngo PL; Steinbeiser MA; Mao SS; Carroll SS; Bailey C; Colussi D; Bosserman M; Burlein C; Cook JJ; Sitko G; Tiller PR; Miller-Stein CM; Rose M; McMasters DR; Vacca JP; Selnick HG Synthesis and evaluation of imidazole acetic acid inhibitors of activated thrombin-activatable fibrinolysis inhibitor as novel antithrombotics. J Med Chem 46:5294-7 (2003) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Carboxypeptidase M | |||
| Name: | Carboxypeptidase M | ||
| Synonyms: | CPM | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 50519.81 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | ChEMBL_45790 | ||
| Residue: | 443 | ||
| Sequence: |
| ||
| BDBM50135939 | |||
| n/a | |||
| Name | BDBM50135939 | ||
| Synonyms: | 3-(4,4-Diamino-but-3-enylsulfanyl)-2-mercaptomethyl-propionic acid | CHEMBL150332 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C8H16N2O2S2 | ||
| Mol. Mass. | 236.355 | ||
| SMILES | NC(=N)CCCSCC(CS)C(O)=O | ||
| Structure | 
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