| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
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| Ligand | BDBM50136798 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200836 (CHEMBL807046) |
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| IC50 | 1.6±n/a nM |
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| Citation |  Erchegyi, J; Waser, B; Schaer, JC; Cescato, R; Brazeau, JF; Rivier, J; Reubi, JC Novel sst(4)-selective somatostatin (SRIF) agonists. 3. Analogues amenable to radiolabeling. J Med Chem46:5597-605 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 4 |
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| Name: | Somatostatin receptor type 4 |
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| Synonyms: | SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42015.38 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P31391 |
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| Residue: | 388 |
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| Sequence: | MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
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| BDBM50136798 |
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| n/a |
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| Name | BDBM50136798 |
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| Synonyms: | CHEMBL410372 | Somatostatin analogue |
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| Type | Small organic molecule |
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| Emp. Form. | C63H75N11O12S2 |
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| Mol. Mass. | 1242.466 |
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| SMILES | C[C@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)C(O)=O)NC(=O)[C@H](N)Cc1ccc(O)cc1 |
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| Structure | 
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