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TargetCalpain small subunit 1
LigandBDBM50137935
Substrate/Competitorn/a
Meas. Tech.ChEBML_43862
Ki>430000±n/a nM
Citation Donkor, IOHan, JZheng, X Design, synthesis, molecular modeling studies, and calpain inhibitory activity of novel alpha-ketoamides incorporating polar residues at the P1'-position. J Med Chem47:72-9 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calpain small subunit 1
Name:Calpain small subunit 1
Synonyms:CANP small subunit | CAPN4 | CAPNS1 | CDPS | CPNS1_PIG | CSS1 | Calcium-activated neutral proteinase small subunit | Calcium-dependent protease small subunit | Calcium-dependent protease small subunit 1 | Calpain regulatory subunit
Type:PROTEIN
Mol. Mass.:28062.13
Organism:Sus scrofa
Description:ChEMBL_43862
Residue:266
Sequence:
MFLVNSFLKGGGGGGGGGGGLGGGLGNVLGGLISGAGGGGGGGGGGGGGGGGGGTAMRIL
GGVISAISEAAAQYNPEPPPPRTHYSNIEANESEEVRQFRRLFAQLAGDDMEVSATELMN
ILNKVVTRHPDLKTDGFGIDTCRSMVAVMDSDTTGKLGFEEFKYLWNNIKKWQAIYKQFD
VDRSGTIGSSELPGAFEAAGFHLNEHLYSMIIRRYSDEGGNMDFDNFISCLVRLDAMFRA
FKSLDKDGTGQIQVNIQEWLQLTMYS
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  Blast E-value cutoff:
BDBM50137935
n/a
NameBDBM50137935
Synonyms:2-[(S)-3-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-4-phenyl-butyrylamino]-3-(R)-phenyl-propionic acid | CHEMBL175176
TypeSmall organic molecule
Emp. Form.C33H37N3O7
Mol. Mass.587.6628
SMILESCC(C)CC(NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(=O)N[C@H](Cc1ccccc1)C(O)=O
Structure
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