Ki Summary new BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetMu-type opioid receptor
LigandBDBM50138007
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145149
Ki 0.07±n/a nM
Citation Zhang AXiong WBidlack JMHilbert JEKnapp BIWentland MPNeumeyer JL 10-Ketomorphinan and 3-substituted-3-desoxymorphinan analogues as mixed kappa and micro opioid ligands: synthesis and biological evaluation of their binding affinity at opioid receptors. J Med Chem 47:165-74 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50138007
n/a
NameBDBM50138007
Synonyms:3-Carboxamido-N-methylmorphinan | CHEMBL297292
TypeSmall organic molecule
Emp. Form.C18H24N2O
Mol. Mass.284.396
SMILESCN1CC[C@]23CCCC[C@H]2[C@H]1Cc1ccc(cc31)C(N)=O
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: