| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipase A2, major isoenzyme |
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| Ligand | BDBM50139530 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_155880 |
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| Ki | 15000±n/a nM |
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| Citation |  Lin, G; Lin, YF; Hwang, MT; Lin, YZ Benzene-di-N-octylcarbamates as conformationally constrained phospholipase A(2) inhibitors. Bioorg Med Chem Lett14:751-5 (2004) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipase A2, major isoenzyme |
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| Name: | Phospholipase A2, major isoenzyme |
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| Synonyms: | Group IB phospholipase A2 | PA21B_PIG | PLA2G1B | Phosphatidylcholine 2-acylhydrolase | Phospholipase A2 |
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| Type: | Hydrolase; monomer or homodimer |
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| Mol. Mass.: | 16279.83 |
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| Organism: | Sus scrofa (pig) |
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| Description: | Purchased from Sigma. |
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| Residue: | 146 |
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| Sequence: | MKFLVLAVLLTVGAAQEGISSRALWQFRSMIKCAIPGSHPLMDFNNYGCYCGLGGSGTPV
DELDRCCETHDNCYRDAKNLDSCKFLVDNPYTESYSYSCSNTEITCNSKNNACEAFICNC
DRNAAICFSKAPYNKEHKNLDTKKYC
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| BDBM50139530 |
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| n/a |
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| Name | BDBM50139530 |
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| Synonyms: | CHEMBL434865 | Octyl-carbamic acid 4-octylcarbamoyloxy-phenyl ester |
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| Type | Small organic molecule |
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| Emp. Form. | C24H40N2O4 |
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| Mol. Mass. | 420.5854 |
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| SMILES | CCCCCCCCNC(=O)Oc1ccc(OC(=O)NCCCCCCCC)cc1 |
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| Structure | 
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