Ki Summary

Reaction Details

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Target

Oligopeptide transporter small intestine isoform

Ligand

BDBM50139892

Substrate/Competitor

n/a

Meas. Tech.

ChEMBL_89215

180±n/a nM

Citation

Våbenø J; Lejon T; Nielsen CU; Steffansen B; Chen W; Ouyang H; Borchardt RT; Luthman K Phe-Gly dipeptidomimetics designed for the di-/tripeptide transporters PEPT1 and PEPT2: synthesis and biological investigations. J Med Chem 47:1060-9 (2004) [PubMed] Article

More Info.:

Get all data from this article, Assay Method

Oligopeptide transporter small intestine isoform

Name:

Oligopeptide transporter small intestine isoform

Synonyms:

Intestinal H(+)/peptide cotransporter | Oligopeptide transporter, small intestine isoform | Peptide transporter 1

Type:

PROTEIN

Mol. Mass.:

78818.07

Organism:

Homo sapiens (Human)

Description:

ChEMBL_1488839

Residue:

708

Sequence:

MGMSKSHSFFGYPLSIFFIVVNEFCERFSYYGMRAILILYFTNFISWDDNLSTAIYHTFV
ALCYLTPILGALIADSWLGKFKTIVSLSIVYTIGQAVTSVSSINDLTDHNHDGTPDSLPV
HVVLSLIGLALIALGTGGIKPCVSAFGGDQFEEGQEKQRNRFFSIFYLAINAGSLLSTII
TPMLRVQQCGIHSKQACYPLAFGVPAALMAVALIVFVLGSGMYKKFKPQGNIMGKVAKCI
GFAIKNRFRHRSKAFPKREHWLDWAKEKYDERLISQIKMVTRVMFLYIPLPMFWALFDQQ
GSRWTLQATTMSGKIGALEIQPDQMQTVNAILIVIMVPIFDAVLYPLIAKCGFNFTSLKK
MAVGMVLASMAFVVAAIVQVEIDKTLPVFPKGNEVQIKVLNIGNNTMNISLPGEMVTLGP
MSQTNAFMTFDVNKLTRINISSPGSPVTAVTDDFKQGQRHTLLVWAPNHYQVVKDGLNQK
PEKGENGIRFVNTFNELITITMSGKVYANISSYNASTYQFFPSGIKGFTISSTEIPPQCQ
PNFNTFYLEFGSAYTYIVQRKNDSCPEVKVFEDISANTVNMALQIPQYFLLTCGEVVFSV
TGLEFSYSQAPSNMKSVLQAGWLLTVAVGNIIVLIVAGAGQFSKQWAEYILFAALLLVVC
VIFAIMARFYTYINPAEIEAQFDEDEKKNRLEKSNPYFMSGANSQKQM

BDBM50139892

n/a

Name

BDBM50139892

Synonyms:

(S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propionic acid | (S,S)2-(2-phenyl-1-trimethylammonioethylcarboxamido)propanoate | CHEMBL429950 | Phe-Ala

Type

Small organic molecule

Emp. Form.

C12H16N2O3

Mol. Mass.

236.267

SMILES

C[C@H](NC(=O)[C@@H](N)Cc1ccccc1)C(O)=O

Structure