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TargetMelatonin receptor type 1B
LigandBDBM50142201
Substrate/Competitorn/a
Meas. Tech.ChEBML_105277
Ki 0.780000±n/a nM
Citation Epperson, JRDeskus, JAGentile, AJIben, LGRyan, ESarbin, NS 4-Substituted anilides as selective melatonin MT2 receptor agonists. Bioorg Med Chem Lett14:1023-6 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Melatonin receptor type 1B
Name:Melatonin receptor type 1B
Synonyms:MTNR1B | MTR1B_HUMAN | Mel-1B-R | Mel1b melatonin receptor | Melatonin 1B | Melatonin receptor | Melatonin receptor type 1B | Melatonin receptor type 2 (MT2)
Type:Enzyme
Mol. Mass.:40203.54
Organism:Homo sapiens (Human)
Description:P49286
Residue:362
Sequence:
MSENGSFANCCEAGGWAVRPGWSGAGSARPSRTPRPPWVAPALSAVLIVTTAVDVVGNLL
VILSVLRNRKLRNAGNLFLVSLALADLVVAFYPYPLILVAIFYDGWALGEEHCKASAFVM
GLSVIGSVFNITAIAINRYCYICHSMAYHRIYRRWHTPLHICLIWLLTVVALLPNFFVGS
LEYDPRIYSCTFIQTASTQYTAAVVVIHFLLPIAVVSFCYLRIWVLVLQARRKAKPESRL
CLKPSDLRSFLTMFVVFVIFAICWAPLNCIGLAVAINPQEMAPQIPEGLFVTSYLLAYFN
SCLNAIVYGLLNQNFRREYKRILLALWNPRHCIQDASKGSHAEGLQSPAPPIIGVQHQAD
AL
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  Blast E-value cutoff:
BDBM50142201
n/a
NameBDBM50142201
Synonyms:CHEMBL7875 | N-(4-Benzofuran-4-ylmethyl-phenyl)-butyramide
TypeSmall organic molecule
Emp. Form.C19H19NO2
Mol. Mass.293.3597
SMILESCCCC(=O)Nc1ccc(Cc2cccc3occc23)cc1
Structure
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