| Reaction Details |
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 | Report a problem with these data |
| Target | Melatonin receptor type 1B |
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| Ligand | BDBM50142228 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_105277 |
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| Ki | 0.680000±n/a nM |
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| Citation |  Epperson, JR; Deskus, JA; Gentile, AJ; Iben, LG; Ryan, E; Sarbin, NS 4-Substituted anilides as selective melatonin MT2 receptor agonists. Bioorg Med Chem Lett14:1023-6 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Melatonin receptor type 1B |
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| Name: | Melatonin receptor type 1B |
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| Synonyms: | MTNR1B | MTR1B_HUMAN | Mel-1B-R | Mel1b melatonin receptor | Melatonin 1B | Melatonin receptor | Melatonin receptor type 1B | Melatonin receptor type 2 (MT2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 40203.54 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P49286 |
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| Residue: | 362 |
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| Sequence: | MSENGSFANCCEAGGWAVRPGWSGAGSARPSRTPRPPWVAPALSAVLIVTTAVDVVGNLL
VILSVLRNRKLRNAGNLFLVSLALADLVVAFYPYPLILVAIFYDGWALGEEHCKASAFVM
GLSVIGSVFNITAIAINRYCYICHSMAYHRIYRRWHTPLHICLIWLLTVVALLPNFFVGS
LEYDPRIYSCTFIQTASTQYTAAVVVIHFLLPIAVVSFCYLRIWVLVLQARRKAKPESRL
CLKPSDLRSFLTMFVVFVIFAICWAPLNCIGLAVAINPQEMAPQIPEGLFVTSYLLAYFN
SCLNAIVYGLLNQNFRREYKRILLALWNPRHCIQDASKGSHAEGLQSPAPPIIGVQHQAD
AL
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| BDBM50142228 |
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| n/a |
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| Name | BDBM50142228 |
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| Synonyms: | CHEMBL7700 | N-[4-(2,3-Dihydro-benzofuran-4-yloxy)-phenyl]-butyramide |
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| Type | Small organic molecule |
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| Emp. Form. | C18H19NO3 |
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| Mol. Mass. | 297.3484 |
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| SMILES | CCCC(=O)Nc1ccc(Oc2cccc3OCCc23)cc1 |
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| Structure | 
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