| Reaction Details |
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 | Report a problem with these data |
| Target | Peptide deformylase |
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| Ligand | BDBM50153086 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_303553 (CHEMBL828953) |
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| Ki | 92±n/a nM |
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| Citation |  Hu, X; Nguyen, KT; Jiang, VC; Lofland, D; Moser, HE; Pei, D Macrocyclic inhibitors for peptide deformylase: a structure-activity relationship study of the ring size. J Med Chem47:4941-9 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Peptide deformylase |
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| Name: | Peptide deformylase |
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| Synonyms: | 3.5.1.88 | BON69_24600 | BON94_18585 | D9G11_24945 | D9G11_25760 | D9J60_20755 | FORC82_p394 | PDF | Polypeptide deformylase | SAMEA3472033_04733 | def | def_2 |
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| Type: | n/a |
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| Mol. Mass.: | 16901.39 |
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| Organism: | Escherichia coli |
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| Description: | n/a |
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| Residue: | 150 |
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| Sequence: | MSVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEKGIGLAATQVDIHQRIIV
IDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFE
LEADGLLAICIGLRLGNGKYCTLRLFFNQV
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| BDBM50153086 |
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| n/a |
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| Name | BDBM50153086 |
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| Synonyms: | CHEMBL188671 | N-[(1R,2S)-3-(4-Amino-butyl)-2,5-dioxo-1,4diaza-cyclopentadec-6-ylmethyl]-N-hydroxy-formamide |
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| Type | Small organic molecule |
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| Emp. Form. | C19H36N4O4 |
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| Mol. Mass. | 384.5135 |
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| SMILES | NCCCC[C@@H]1NC(=O)[C@@H](CN(O)C=O)CCCCCCCCCNC1=O |
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| Structure | 
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