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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Trypsin | ||
| Ligand | BDBM50147088 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_302473 | ||
| Ki | 45±n/a nM | ||
| Citation |  Bruncko M; McClellan WJ; Wendt MD; Sauer DR; Geyer A; Dalton CR; Kaminski MA; Weitzberg M; Gong J; Dellaria JF; Mantei R; Zhao X; Nienaber VL; Stewart K; Klinghofer V; Bouska J; Rockway TW; Giranda VL Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties. Bioorg Med Chem Lett 15:93-8 (2004) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Trypsin | |||
| Name: | Trypsin | ||
| Synonyms: | n/a | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 24411.24 | ||
| Organism: | Sus scrofa | ||
| Description: | ChEMBL_1450738 | ||
| Residue: | 231 | ||
| Sequence: |
| ||
| BDBM50147088 | |||
| n/a | |||
| Name | BDBM50147088 | ||
| Synonyms: | 6-Carbamimidoyl-4-furan-3-yl-naphthalene-2-carboxylic acid phenylamide | CHEMBL319047 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C22H17N3O2 | ||
| Mol. Mass. | 355.3893 | ||
| SMILES | NC(=N)c1ccc2cc(cc(-c3ccoc3)c2c1)C(=O)Nc1ccccc1 | ||
| Structure | 
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