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TargetGag-Pol polyprotein [489-587]
LigandBDBM50157216
Substrate/Competitorn/a
Meas. Tech.ChEMBL_305393 (CHEMBL833043)
IC50 10000±n/a nM
Citation Garino, CBihel, FPietrancosta, NLaras, YQuéléver, GWoo, IKlein, PBain, JBoucher, JLKraus, JL New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties. Bioorg Med Chem Lett15:135-8 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Gag-Pol polyprotein [489-587]
Name:Gag-Pol polyprotein [489-587]
Synonyms:Human immunodeficiency virus type 1 protease | POL_HV1H2 | Pol polyprotein | gag-pol
Type:Enzyme Subunit
Mol. Mass.:10781.16
Organism:Human immunodeficiency virus type 1
Description:P04585[489-587]
Residue:99
Sequence:
PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYD
QILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF
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BDBM50157216
n/a
NameBDBM50157216
Synonyms:2-Bromomethyl-8-nitro-benzo[c]chromen-6-one | CHEMBL369126
TypeSmall organic molecule
Emp. Form.C14H8BrNO4
Mol. Mass.334.122
SMILES[O-][N+](=O)c1ccc2c3cc(CBr)ccc3oc(=O)c2c1
Structure
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