| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
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| Ligand | BDBM50166114 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_304392 (CHEMBL830042) |
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| EC50 | >10000±n/a nM |
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| Citation |  Xu, Y; Aoki, J; Shimizu, K; Umezu-Goto, M; Hama, K; Takanezawa, Y; Yu, S; Mills, GB; Arai, H; Qian, L; Prestwich, GD Structure-activity relationships of fluorinated lysophosphatidic acid analogues. J Med Chem48:3319-27 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 3 |
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| Name: | Lysophosphatidic acid receptor 3 |
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| Synonyms: | EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7 |
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| Type: | Enzyme |
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| Mol. Mass.: | 40149.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9UBY5 |
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| Residue: | 353 |
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| Sequence: | MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
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| BDBM50166114 |
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| n/a |
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| Name | BDBM50166114 |
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| Synonyms: | (E)-Octadec-9-enoic acid (S)-3,3-difluoro-1-phosphonooxymethyl-allyl ester | CHEMBL191737 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H41F2O6P |
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| Mol. Mass. | 470.5279 |
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| SMILES | CCCCCCCC\C=C\CCCCCCCC(=O)O[C@H](COP(O)(O)=O)CC(F)F |
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| Structure | 
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