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TargetLysophosphatidic acid receptor 3
LigandBDBM50170852
Substrate/Competitorn/a
Meas. Tech.ChEMBL_303206 (CHEMBL829832)
Ki 14±n/a nM
Citation Durgam, GGVirag, TWalker, MDTsukahara, RYasuda, SLiliom, Kvan Meeteren, LAMoolenaar, WHWilke, NSiess, WTigyi, GMiller, DD Synthesis, structure-activity relationships, and biological evaluation of fatty alcohol phosphates as lysophosphatidic acid receptor ligands, activators of PPARgamma, and inhibitors of autotaxin. J Med Chem48:4919-30 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lysophosphatidic acid receptor 3
Name:Lysophosphatidic acid receptor 3
Synonyms:EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7
Type:Enzyme
Mol. Mass.:40149.72
Organism:Homo sapiens (Human)
Description:Q9UBY5
Residue:353
Sequence:
MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
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  Blast E-value cutoff:
BDBM50170852
n/a
NameBDBM50170852
Synonyms:CHEMBL187402 | Thiophosphoric acid (E)-tetradec-9-enyl ester
TypeSmall organic molecule
Emp. Form.C14H29O3PS
Mol. Mass.308.417
SMILESCCCC\C=C\CCCCCCCCOP(O)(O)=S
Structure
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