| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
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| Ligand | BDBM50176396 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_333864 (CHEMBL865902) |
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| IC50 | 414±n/a nM |
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| Citation |  Durgam, GG; Tsukahara, R; Makarova, N; Walker, MD; Fujiwara, Y; Pigg, KR; Baker, DL; Sardar, VM; Parrill, AL; Tigyi, G; Miller, DD Synthesis and pharmacological evaluation of second-generation phosphatidic acid derivatives as lysophosphatidic acid receptor ligands. Bioorg Med Chem Lett16:633-40 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 3 |
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| Name: | Lysophosphatidic acid receptor 3 |
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| Synonyms: | EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7 |
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| Type: | Enzyme |
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| Mol. Mass.: | 40149.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9UBY5 |
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| Residue: | 353 |
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| Sequence: | MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
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| BDBM50176396 |
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| n/a |
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| Name | BDBM50176396 |
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| Synonyms: | CHEMBL204037 | Serine amide phospate derivative | phosphoric acid mono-((S)-2-octanoylamino-2-octylcarbamoyl-ethyl) ester |
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| Type | Small organic molecule |
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| Emp. Form. | C19H39N2O6P |
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| Mol. Mass. | 422.4965 |
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| SMILES | CCCCCCCCNC(=O)[C@H](COP(O)(O)=O)NC(=O)CCCCCCC |
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| Structure | 
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