| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
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| Ligand | BDBM50177334 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_329846 (CHEMBL862795) |
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| EC50 | 692±n/a nM |
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| Citation |  Gududuru, V; Zeng, K; Tsukahara, R; Makarova, N; Fujiwara, Y; Pigg, KR; Baker, DL; Tigyi, G; Miller, DD Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. Bioorg Med Chem Lett16:451-6 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 3 |
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| Name: | Lysophosphatidic acid receptor 3 |
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| Synonyms: | Edg7 | LPAR3_RAT | Lpa3 | Lpar3 | Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3 | Lysophosphatidic acid receptor Edg-7 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40307.81 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_329846 |
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| Residue: | 354 |
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| Sequence: | MNECHYDKRMDFFYNRSNTDTADEWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVITNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWLLRQGLLDTSLTASLANL
LVIAVERHMSIMRMRIHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLIFWTVSNLLAFFIMVVVYVRIYMYVKRKTNVLSPHTSGSISRRRAPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCKQCNVQHVKRWFLLLALLNSVMNPIIYSYKDEDM
YNTMRKMICCAPHDSNAERHPSRIPSTIHSRSDTGSQYLEDSISQGQVCNKSSS
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| BDBM50177334 |
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| n/a |
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| Name | BDBM50177334 |
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| Synonyms: | CHEMBL198406 | potassium O-(2-(6-(4-octylphenyl)hexyl)-1,3-dioxolan-4-yl)methyl O-hydrogenphosphorothioate |
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| Type | Small organic molecule |
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| Emp. Form. | C24H40O5PS |
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| Mol. Mass. | 471.611 |
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| SMILES | CCCCCCCCc1ccc(CCCCCCC2OCC(COP(O)([O-])=S)O2)cc1 |
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| Structure | 
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