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TargetLysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3
LigandBDBM50177329
Substrate/Competitorn/a
Meas. Tech.ChEMBL_329846
Ki 171±n/a nM
Citation Gududuru VZeng KTsukahara RMakarova NFujiwara YPigg KRBaker DLTigyi GMiller DD Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. Bioorg Med Chem Lett 16:451-6 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3
Name:Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3
Synonyms:Lysophosphatidic acid receptor Edg-7
Type:PROTEIN
Mol. Mass.:40307.81
Organism:Rattus norvegicus
Description:ChEMBL_329846
Residue:354
Sequence:
MNECHYDKRMDFFYNRSNTDTADEWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVITNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWLLRQGLLDTSLTASLANL
LVIAVERHMSIMRMRIHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLIFWTVSNLLAFFIMVVVYVRIYMYVKRKTNVLSPHTSGSISRRRAPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCKQCNVQHVKRWFLLLALLNSVMNPIIYSYKDEDM
YNTMRKMICCAPHDSNAERHPSRIPSTIHSRSDTGSQYLEDSISQGQVCNKSSS
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  Blast E-value cutoff:
BDBM50177329
n/a
NameBDBM50177329
Synonyms:CHEMBL199380 | potassium (2-(6-(4-octylphenyl)hexyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate
TypeSmall organic molecule
Emp. Form.C24H40O6P
Mol. Mass.455.5451
SMILESCCCCCCCCc1ccc(CCCCCCC2OCC(COP(O)([O-])=O)O2)cc1
Structure
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