Reaction Details |
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Target | Neuropeptide Y receptor type 2 |
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Ligand | BDBM50197025 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_453177 (CHEMBL902327) |
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Ki | 0.4±n/a nM |
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Citation | DeCarr, LB; Buckholz, TM; Coish, PD; Fathi, Z; Fisk, SE; Mays, MR; O'Connor, SJ; Lumb, KJ Identification of selective neuropeptide Y2 peptide agonists. Bioorg Med Chem Lett17:538-41 (2007) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Neuropeptide Y receptor type 2 |
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Name: | Neuropeptide Y receptor type 2 |
Synonyms: | NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 42734.65 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y2 NPY2R HUMAN::P49146 |
Residue: | 381 |
Sequence: | MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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BDBM50197025 |
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n/a |
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Name | BDBM50197025 |
Synonyms: | CHEMBL439904 | PYY(3-36) |
Type | Small organic molecule |
Emp. Form. | C180H279N53O54 |
Mol. Mass. | 4049.464 |
SMILES | n/a |
Structure |
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