| Reaction Details |
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 | Report a problem with these data |
| Target | Cholecystokinin receptor type A |
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| Ligand | BDBM50208418 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_443246 (CHEMBL893496) |
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| IC50 | 197±n/a nM |
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| Citation |  Tiwari, AK; Mishra, AK; Bajpai, A; Mishra, P; Singh, S; Sinha, D; Singh, VK Synthesis and evaluation of novel benzimidazole derivative [Bz-Im] and its radio/biological studies. Bioorg Med Chem Lett17:2749-55 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cholecystokinin receptor type A |
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| Name: | Cholecystokinin receptor type A |
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| Synonyms: | CCKAR_RAT | Cckar | Cholecystokinin peripheral | Cholecystokinin receptor | Cholecystokinin receptor type A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 49676.37 |
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| Organism: | RAT |
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| Description: | Cholecystokinin central 0 RAT::P30551 |
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| Residue: | 444 |
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| Sequence: | MSHSPARQHLVESSRMDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSALQI
LLYSIIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLK
DFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAAT
WCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLLPGIVM
VVAYGLISLELYQGIKFDASQKKSAKEKKPSTGSSTRYEDSDGCYLQKSRPPRKLELQQL
SSGSGGSRLNRIRSSSSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAE
KHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPPGVRGEVGEEE
DGRTIRALLSRYSYSHMSTSAPPP
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| BDBM50208418 |
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| n/a |
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| Name | BDBM50208418 |
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| Synonyms: | 2-[5-((E)-2-biphenyl-4-yl-vinyl)-2-hydroxy-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl]-isoindole-1,3-dione | CHEMBL233457 | VL-0494 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H25N3O3 |
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| Mol. Mass. | 571.6234 |
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| SMILES | Oc1ccc2c(\C=C\c3ccc(cc3)-c3ccccc3)cc3nc4ccccc4n3c2c1CN1C(=O)c2ccccc2C1=O |
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| Structure | 
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