| Reaction Details |
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 | Report a problem with these data |
| Target | Cholecystokinin receptor type A |
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| Ligand | BDBM50208419 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_443247 (CHEMBL893497) |
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| IC50 | 2940±n/a nM |
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| Citation |  Tiwari, AK; Mishra, AK; Bajpai, A; Mishra, P; Singh, S; Sinha, D; Singh, VK Synthesis and evaluation of novel benzimidazole derivative [Bz-Im] and its radio/biological studies. Bioorg Med Chem Lett17:2749-55 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cholecystokinin receptor type A |
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| Name: | Cholecystokinin receptor type A |
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| Synonyms: | CCK-A receptor | CCK-AR | CCK1-R | CCKAR | CCKAR_CAVPO | Cholecystokinin A receptor | Cholecystokinin receptor type A | Cholecystokinin-1 receptor |
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| Type: | n/a |
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| Mol. Mass.: | 48229.77 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 430 |
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| Sequence: | MDVVDSLFVNGSNITSACELGFENETLFCLDRPRPSKEWQPAVQILLYSLIFLLSVLGNT
LVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPSLLKDFIFGSAVCKTTTYF
MGTSVSVSTFNLVAISLERYGAICKPLQSRVWQTKSHALKVIAATWCLSFTIMTPYPIYS
NLVPFTKNNNQTGNMCRFLLPNDVMQQTWHTFLLLILFLIPGIVMMVAYGLISLELYQGI
KFDAIQKKSAKERKTSTGSSGPMEDSDGCYLQKSRHPRKLELRQLSPSSSGSNRINRIRS
SSSTANLMAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAERHLSGTPISFILLL
SYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGTPGVRGEMGEEEEGRTTGASLSRYSY
SHMSTSAPPP
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| BDBM50208419 |
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| n/a |
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| Name | BDBM50208419 |
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| Synonyms: | 2-{2-hydroxy-5-[(E)-2-(4-hydroxy-phenyl)-vinyl]-benzo[4,5]imidazo[1,2-a]quinolin-1-ylmethyl}-isoindole-1,3-dione | CHEMBL389311 |
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| Type | Small organic molecule |
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| Emp. Form. | C32H21N3O4 |
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| Mol. Mass. | 511.5268 |
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| SMILES | Oc1ccc(\C=C\c2cc3nc4ccccc4n3c3c(CN4C(=O)c5ccccc5C4=O)c(O)ccc23)cc1 |
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| Structure | 
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