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TargetFatty acid-binding protein, heart
LigandBDBM50212880
Substrate/Competitorn/a
Meas. Tech.ChEMBL_455934 (CHEMBL887935)
Ki>1000±n/a nM
Citation Sulsky, RMagnin, DRHuang, YSimpkins, LTaunk, PPatel, MZhu, YStouch, TRBassolino-Klimas, DParker, RHarrity, TStoffel, RTaylor, DSLavoie, TBKish, KJacobson, BLSheriff, SAdam, LPEwing, WRRobl, JA Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). Bioorg Med Chem Lett17:3511-5 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, heart
Name:Fatty acid-binding protein, heart
Synonyms:FABP11 | FABP3 | FABPH_HUMAN | Fatty acid binding protein muscle | MDGI
Type:PROTEIN
Mol. Mass.:14858.36
Organism:Homo sapiens (Human)
Description:ChEMBL_1463784
Residue:133
Sequence:
MVDAFLGTWKLVDSKNFDDYMKSLGVGFATRQVASMTKPTTIIEKNGDILTLKTHSTFKN
TEISFKLGVEFDETTADDRKVKSIVTLDGGKLVHLQKWDGQETTLVRELIDGKLILTLTH
GTAVCTRTYEKEA
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  Blast E-value cutoff:
BDBM50212880
n/a
NameBDBM50212880
Synonyms:CHEMBL245857 | [2'-(1-isobutyl-4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-ylamino]-acetic acid
TypeSmall organic molecule
Emp. Form.C33H31N3O2
Mol. Mass.501.6181
SMILESCC(C)Cn1c(nc(c1-c1ccccc1)-c1ccccc1)-c1ccccc1-c1cccc(NCC(O)=O)c1
Structure
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