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TargetFatty acid-binding protein, adipocyte
LigandBDBM50002838
Substrate/Competitorn/a
Meas. Tech.ChEMBL_455933 (CHEMBL887934)
Ki 58±n/a nM
Citation Sulsky, RMagnin, DRHuang, YSimpkins, LTaunk, PPatel, MZhu, YStouch, TRBassolino-Klimas, DParker, RHarrity, TStoffel, RTaylor, DSLavoie, TBKish, KJacobson, BLSheriff, SAdam, LPEwing, WRRobl, JA Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). Bioorg Med Chem Lett17:3511-5 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, adipocyte
Name:Fatty acid-binding protein, adipocyte
Synonyms:A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | FABP4 | FABP4_HUMAN | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4 | Fatty acid-binding protein 4 (FABP4)
Type:Enzyme
Mol. Mass.:14719.23
Organism:Homo sapiens (Human)
Description:P15090
Residue:132
Sequence:
MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKN
TEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVM
KGVTSTRVYERA
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  Blast E-value cutoff:
BDBM50002838
n/a
NameBDBM50002838
Synonyms:5-(2-(4,5-diphenyloxazol-2-yl)phenoxy)pentanoic acid | 5-[2-(4,5-Diphenyl-oxazol-2-yl)-phenoxy]-pentanoic acid | 5-[2-(4,5-Diphenyl-oxazol-2-yl)-phenoxy]-pentanoic acid;hydrate | CHEMBL116533
TypeSmall organic molecule
Emp. Form.C26H23NO4
Mol. Mass.413.4651
SMILESOC(=O)CCCCOc1ccccc1-c1nc(c(o1)-c1ccccc1)-c1ccccc1
Structure
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