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TargetFatty acid-binding protein 5
LigandBDBM50212881
Substrate/Competitorn/a
Meas. Tech.ChEMBL_455935 (CHEMBL887936)
Ki 830±n/a nM
Citation Sulsky, RMagnin, DRHuang, YSimpkins, LTaunk, PPatel, MZhu, YStouch, TRBassolino-Klimas, DParker, RHarrity, TStoffel, RTaylor, DSLavoie, TBKish, KJacobson, BLSheriff, SAdam, LPEwing, WRRobl, JA Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). Bioorg Med Chem Lett17:3511-5 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein 5
Name:Fatty acid-binding protein 5
Synonyms:FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5)
Type:Enzyme
Mol. Mass.:15164.79
Organism:Homo sapiens (Human)
Description:Q01469
Residue:135
Sequence:
MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
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BDBM50212881
n/a
NameBDBM50212881
Synonyms:CHEMBL396698 | [2'-(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)-biphenyl-3-yloxy]-acetic acid
TypeSmall organic molecule
Emp. Form.C30H24N2O3
Mol. Mass.460.5232
SMILESCn1c(nc(c1-c1ccccc1)-c1ccccc1)-c1ccccc1-c1cccc(OCC(O)=O)c1
Structure
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