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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Motilin receptor | ||
| Ligand | BDBM50214255 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_447562 (CHEMBL896576) | ||
| Ki | 17±n/a nM | ||
| Citation |  Marsault, E; Benakli, K; Beaubien, S; Saint-Louis, C; Déziel, R; Fraser, G Potent macrocyclic antagonists to the motilin receptor presenting novel unnatural amino acids. Bioorg Med Chem Lett17:4187-90 (2007) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Motilin receptor | |||
| Name: | Motilin receptor | ||
| Synonyms: | G-protein coupled receptor 38 | GPR38 | MLNR | MTLR | MTLR1 | MTLR_HUMAN | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 45365.95 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | ChEMBL_122664 | ||
| Residue: | 412 | ||
| Sequence: |
| ||
| BDBM50214255 | |||
| n/a | |||
| Name | BDBM50214255 | ||
| Synonyms: | (5R,8R,11S)-11-[(5-methyl-1H-1,2,3-triazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione | CHEMBL269007 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C32H40F3N7O4 | ||
| Mol. Mass. | 643.6997 | ||
| SMILES | CC(C)[C@H]1NC(=O)[C@@H](Cc2cccc(c2)C(F)(F)F)NCCOc2ccccc2CCCNC(=O)[C@H](Cn2nncc2C)NC1=O | ||
| Structure | 
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