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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50217008
Substrate/Competitorn/a
Meas. Tech.ChEMBL_440343 (CHEMBL890658)
Ki 6±n/a nM
Citation Pham, TQGreguric, ILiu, XBerghofer, PBallantyne, PChapman, JMattner, FDikic, BJackson, TLoc'h, CKatsifis, A Synthesis and evaluation of novel radioiodinated benzamides for malignant melanoma. J Med Chem50:3561-72 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:OPRS1 | SGMR1_CAVPO | SIGMAR1 | Sigma 1-type opioid receptor | Sigma non-opioid intracellular receptor 1 | Sigma-1 receptor | Sigma1-receptor | Sigma1R | Sterol isomerase-like protein
Type:Protein
Mol. Mass.:25307.17
Organism:Cavia porcellus (Guinea pig)
Description:Q60492
Residue:223
Sequence:
MQWAVGRRWLWVALFLAAVAVLTQIVWLWLGTQNFVFQREEIAQLARQYAGLDHELAFSK
LIVELRRLHPVHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSPRHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLGFALADTVFSTQDFLTLFYTLRVYARALQLELTTYLFGQDP
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BDBM50217008
n/a
NameBDBM50217008
Synonyms:CHEMBL230904 | N-(1-(2-fluoroethyl)piperidin-4-yl)-4-iodobenzamide
TypeSmall organic molecule
Emp. Form.C15H21FIN3O
Mol. Mass.405.2496
SMILESFCCN1CCN(CCNC(=O)c2ccc(I)cc2)CC1
Structure
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