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TargetCarboxypeptidase B
LigandBDBM50201438
Substrate/Competitorn/a
Meas. Tech.ChEMBL_452075
Ki 0.420000±n/a nM
Citation Bunnage MEBlagg JSteele JOwen DRAllerton CMcElroy ABMiller DRinger TButcher KBeaumont KEvans KGray AJHolland SJFeeder NMoore RSBrown DG Discovery of potent& selective inhibitors of activated thrombin-activatable fibrinolysis inhibitor for the treatment of thrombosis. J Med Chem 50:6095-103 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Carboxypeptidase B
Name:Carboxypeptidase B
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:47371.10
Organism:Sus scrofa
Description:ChEMBL_453905
Residue:416
Sequence:
MLAFLILVTVTLASAHHSGEHFEGEKVFRVNVEDENDISLLHELASTRQIDFWKPDSVTQ
IKPHSTVDFRVKAEDILAVEDFLEQNELQYEVLINNLRSVLEAQFDSRVRTTGHSYEKYN
NWETIEAWTKQVTSENPDLISRTAIGTTFLGNNIYLLKVGKPGPNKPAIFMDCGFHAREW
ISHAFCQWFVREAVLTYGYESHMTEFLNKLDFYVLPVLNIDGYIYTWTKNRMWRKTRSTN
AGTTCIGTDPNRNFDAGWCTTGASTDPCDETYCGSAAESEKETKALADFIRNNLSSIKAY
LTIHSYSQMILYPYSYDYKLPENNAELNNLAKAAVKELATLYGTKYTYGPGATTIYPAAG
GSDDWAYDQGIKYSFTFELRDKGRYGFILPESQIQATCEETMLAIKYVTNYVLGHL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50201438
n/a
NameBDBM50201438
Synonyms:(+/-)-5-guanidino-2-(mercaptomethyl)pentanoic acid | 5-guanidino-2-(mercaptomethyl)pentanoic acid | CHEMBL236822
TypeSmall organic molecule
Emp. Form.C7H15N3O2S
Mol. Mass.205.278
SMILES[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6](-[#6]-[#16])-[#6](-[#8])=O
Structure
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