| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50242566 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_534563 (CHEMBL988124) |
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| IC50 | 4820±n/a nM |
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| Citation |  Song, KS; Lee, SH; Chun, HJ; Kim, JY; Jung, ME; Ahn, K; Kim, SU; Kim, J; Lee, J Design, synthesis and biological evaluation of piperazine analogues as CB1 cannabinoid receptor ligands. Bioorg Med Chem16:4035-51 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50242566 |
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| n/a |
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| Name | BDBM50242566 |
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| Synonyms: | CHEMBL519584 | N-tert-Butyl-4-((2-chlorophenyl)(4-chlorophenyl)-methyl)piperazine-1-carboxamide |
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| Type | Small organic molecule |
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| Emp. Form. | C22H27Cl2N3O |
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| Mol. Mass. | 420.375 |
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| SMILES | CC(C)(C)NC(=O)N1CCN(CC1)C(c1ccc(Cl)cc1)c1ccccc1Cl |
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| Structure | 
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