| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM50251331 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_533454 (CHEMBL986946) |
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| Ki | >10000±n/a nM |
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| Citation |  Sipos, A; Csutorás, C; Berényi, S; Uustare, A; Rinken, A Synthesis and neuropharmacological characterization of 2-O-substituted apomorphines. Bioorg Med Chem16:4563-8 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | D(1A) dopamine receptor | DOPAMINE D1 | DRD1_MOUSE | Dopamine D1 receptor | Dopamine receptor | Drd1 | Drd1a | Gpcr15 |
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| Type: | Enzyme |
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| Mol. Mass.: | 49613.93 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | Q61616 |
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| Residue: | 446 |
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| Sequence: | MAPNTSTMDETGLPVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNF
FVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDR
YWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLED
AEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKN
CQTTTGNGNPVECSQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGS
EETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIET
VSINNNGAVMFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKREEAGGIPKPLEKLSPAL
SVILDYDTDVSLEKIQPVTHSGQHST
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| BDBM50251331 |
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| n/a |
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| Name | BDBM50251331 |
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| Synonyms: | Bis-{[R-(-)-apomorphine-2-oxy]ethyl} ether | CHEMBL444149 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H40N2O7 |
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| Mol. Mass. | 636.7334 |
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| SMILES | CN1CCc2cc(OCCOCCOc3cc4CCN(C)[C@@H]5Cc6ccc(O)c(O)c6-c(c3)c45)cc-3c2[C@H]1Cc1ccc(O)c(O)c-31 |r| |
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| Structure | 
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