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TargetGlutathione transferase
LigandBDBM50227631
Substrate/Competitorn/a
Meas. Tech.ChEMBL_553571 (CHEMBL958754)
IC50 0.900000±n/a nM
Citation Friesen, RWMancini, JA Microsomal prostaglandin E2 synthase-1 (mPGES-1): a novel anti-inflammatory therapeutic target. J Med Chem51:4059-67 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Glutathione transferase
Name:Glutathione transferase
Synonyms:Microsomal prostaglandin E synthase-1
Type:PROTEIN
Mol. Mass.:17345.98
Organism:Sus scrofa
Description:ChEMBL_553571
Residue:153
Sequence:
MPPPSLEMVSGQVLPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDAQRHGGLQYC
RSDPDVERCLRAHRNDMETIYPFLFLGLVYSFLGPDPFVAWMHFLIFFLGRMVHTIAYLG
KLRAPTRSLAYTLAQLPCASMALQIVWEAARHL
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  Blast E-value cutoff:
BDBM50227631
n/a
NameBDBM50227631
Synonyms:2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile | CHEMBL412099
TypeSmall organic molecule
Emp. Form.C23H11ClN4
Mol. Mass.378.813
SMILESClc1ccc2c3[nH]c(nc3c3ccccc3c2c1)-c1c(cccc1C#N)C#N
Structure
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