| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50271441 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_556845 (CHEMBL964705) |
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| IC50 | 64.41±n/a nM |
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| Citation |  Wang, CL; Yao, JL; Yu, Y; Shao, X; Cui, Y; Liu, HM; Lai, LH; Wang, R Structure-activity study of endomorphin-2 analogs with C-terminal modifications by NMR spectroscopy and molecular modeling. Bioorg Med Chem16:6415-22 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | Mu-opioid receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 44729.40 |
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| Organism: | Cavia porcellus |
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| Description: | ChEMBL_510437 |
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| Residue: | 400 |
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| Sequence: | MDSGAVPGNASDCTDPFAQSTCSPAPSPGSWTNLSHLDGNLSDPCGPNRTDLVGSDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIVNVCNWILSSAIGLPVMFMATTKYRNGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALITIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSTI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM50271441 |
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| n/a |
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| Name | BDBM50271441 |
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| Synonyms: | CHEMBL505502 | Tyr-Pro-Phe-Phe-OCH2CH3 |
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| Type | Small organic molecule |
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| Emp. Form. | C34H40N4O6 |
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| Mol. Mass. | 600.7046 |
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| SMILES | CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1 |r| |
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| Structure | 
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